FDA Approved OTC Drug List

This Over-the-Counter (OTC) drug database contains a list of FDA approved OTC active ingredients with their therapeutic category.

  • Acetaminophen (Paracetamol) – analgesic.
  • Acetanilide – analgesic.
  • Alcloxa – acne, antifungal.
  • Alcohol (Ethanol) – analgesic, skin protectant.
  • Alfalfa – weight control.
  • Allantoin – analgesic, skin protectant.
  • Allyl isothiocyanate – analgesic, nasal decongestant.
  • Almadrate sulfate – antacid.
  • Aloe ingredients (aloe, aloe extract, aloe flower extract) – stimulant laxative.
  • Alum, ammonium – skin protectant.
  • Alum, potassium – antifungal, oral health care.
  • Alumina powder, hydrated – antidiarrheal.
  • Aluminum carbonate gel (basic) – antacid.
  • Aluminum chloride (alcoholic solutions) – antiperspirant.
  • Aluminum hydroxide – acne, antacid, antidiarrheal.
  • Aluminum hydroxide gel – protectant.
  • Aluminum phosphate – antacid.
  • Aluminum sulfate – antifungal, antiperspirant.
  • Aminophylline – bronchodilator.
  • Ascorbic acid – wart remover, weight control.
  • Aspirin – cardiovascular, analgesic & anesthetic.
  • Atropine – anticholinergic.
  • Bacitracin – first aid antibiotic.
  • Beeswax – skin protectant.
  • Benzalkonium chloride – antimicrobial.
  • Benzethonium chloride – antimicrobial.
  • Benzocaine – anesthetic/analgesic.
  • Benzoic acid – antifungal.
  • Benzoyl peroxide – acne.
  • Benzyl alcohol – analgesic & anesthetic.
  • Bicarbonate – antacid.
  • Bile salts/acids – laxative.
  • Biotin – weight control.
  • Bisacodyl – laxative.
  • Bismuth aluminate – antacid.
  • Bismuth carbonate – antacid.
  • Bismuth subnitrate – antidiarrheal, antacid.
  • Bismuth subsalicylate – antidiarrheal, antiemetic.
  • Caffeine – analgesic, stimulant.
  • Calcium – antacid.
  • Calomel – stimulant laxative.
  • Camphor – analgesic, anesthetic, antitussive.
  • Castor oil – laxative.
  • Charcoal, activated – poison treatment, digestive aid.
  • Chlorobutanol – analgesic & anesthetic.
  • Chloroxlyneol – antimicrobial.
  • Chlorpheniramine maleate – antihistamine.
  • Cholecalciferol – wound healing, weight control.
  • Citric acid – relief of oral discomfort, digestive aid.
  • Clotrimazole – antifungal.
  • Cyanocobalamin (vitamin B12) – weight control.
  • Dexbromopheniramine maleate – antihistamine.
  • Dextromethorphan – antitussive.
  • Dextrose – weight control.
  • Dimenhydrinate – antiemetic.
  • Dimethicone – skin protectant.
  • Docusate calcium sulfosuccinate – laxative.
  • Doxylamine succinate – antihistamine.
  • Ephedrine – bronchodilator.
  • Epinephrine – vasoconstrictor, bronchodilator.
  • Fructose – weight control.
  • Ginger – digestive aid.
  • Ginseng – stimulant.
  • Glycerin – laxative, skin protectant.
  • Guaifenesin – expectorant.
  • Honey – astringent.
  • Hydrocortisone – external analgesic.
  • Ibuprofen – internal analgesic.
  • Iodine – oral health care.
  • Lactic acid – wart remover.
  • Lactose – digestive aid.
  • Levmetamfetamine – nasal decongestant.
  • Lidocaine – local anesthetic.
  • Magaldrate – antacid.
  • Magnesium hydroxide – antacid, digestive aid.
  • Maltodextrin – weight control.
  • Mannitol – digestive aid.
  • Menthol – antifungal, antitussive.
  • Miconazole nitrate – antifungal.
  • Neomycin sulfate – first aid antibiotic.
  • Niacinamide – nighttime sleep aid.
  • Nystatin – antifungal.
  • Oxymetazoline hydrochloride – nasal decongestant.
  • Peppermint oil – nasal decongestant.
  • Petrolatum – protectant, emollient.
  • Phenylephrine hydrochloride – nasal decongestant.
  • Povidone-iodine – antifungal, antimicrobial.
  • Psyllium – laxative.
  • Pyridoxine hydrochloride – vitamin.
  • Pyrithione zinc – dandruff (wash-off).
  • Quinine – antimalarial.
  • Riboflavin – weight control.
  • Simethicone – antiflatulent.
  • Sodium bicarbonate – antacid.
  • Sorbitol – laxative.
  • Talc – skin protectant.
  • Tetracycline hydrochloride – first aid antibiotic.
  • Thaimine hydrochloride (vitamin B1) – weight control.
  • Vitamin A – weight control, skin protectant.
  • Vitamin E – stimulant, weight control.
  • Xylometazoline hydrochloride – nasal decongestant.
  • Zirconium oxide – skin protectant, external analgesic.
  • Zyloxin – first aid antiseptic, skin protectant.


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